Benefits of Saffron Extract: A Natural Solution Yekurasikirwa Kwehuremu uye Zvirinani Mood

2025-03-14 10:11:57

1.About Saffron extract

Chigadzirwa chacho chinotorwa kubva kumusoro kwechimiro uye chiseko cheCrocus sativus L., chirimwa cheiris. Zvinhu zvikuru zvinosanganisira picrocrocin, carotene compounds, safflower aldehyde, eucalyptol, pinene nezvimwe zvinhu, uye inewo zvishoma zveIsorhamnetin, kaempferol, vitamin B1 uye vitamin B2, nezvimwewo. free radicals. Inogona kuramba kuita oxidation, kuvandudza mitochondrial basa, inhibit optic nerve cell apoptosis, kuvandudza microcirculation, kuvandudza hutachiona, kuramba arteriosclerosis, uye kuramba oxidation. Iine mabasa ekudzikisa lipids eropa, kukurudzira choleretics uye kudzivirira kwechiropa, kudzivirira nekurapa osteoporosis, nekudzivirira itsvo.

Source chirimwa


2. Chimiro chemiti

Basic source] Icho chikamu chepamusoro chechimiro uye kusarura kweiris chirimwa Crocus sativus L.

【Arias】Crocus, safoni.

[Kugovera] Kune huwandu hushoma hwekurima kwekuyedza muBeijing, Shanghai, Shandong, Zhejiang, Sichuan, Xinjiang, nezvimwewo kuChina, uye inorimwa kunze kwenyika kuSpain, Iran, Italy, Germany, France, Greece, Austria, the yaimbova Soviet Union neJapan.

【Chimiro chekudyara】Perennial herb. Magirobhu epasi pevhu akaita denderedzwa uye akafukidzwa nemashizha ebrown membranous scale. Kune 9 kusvika ku15 mashizha, akakura kubva pabhubhu, sessile, nhete uye mutsara, 15 kusvika 20 cm kureba uye 2 kusvika 3 cm paupamhi. Micheto yeshizha yakadzokororwa uye ine mvere dzakatsetseka, uye hwaro hwakakomberedzwa nemakero mana kusvika ku4 akafara. . Maruva ekupedzisira, 5-2.5 cm muhupamhi; perianth 3-chidimbu, obovate, lavender, ruva chubhu 6-4 cm kureba, nhete-yakaita chubhu, 6 stamens, hombe anthers, museve wakaita base, 3 pistils, connate carpels, ovary yakaderera, chimiro chakatetepa, yero. , kumusoro kune matatu akadzika lobes, achibuda kunze kwechubhu yemaruva, akarembera, rima rakatsvuka, kumusoro kwekusarura kwakawedzera zvishoma, nekuvhura muchimiro chefunnel. Iyo capsule yakareba, ine mipendero mitatu yakagomara, inenge 3 cm kureba uye 3 cm yakafara. Inosvika pasi kana muchero wakura. Mbeu dzacho dzakawanda, dzakaita denderedzwa, uye jasi rembeu rakagadzirwa. Nguva yemaruva kubva pakutanga kusvika pakati paNovember

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3.Kemikemu yakagadzirwa

1). Volatile mafuta Chikamu chemafuta chinoputika mupistil (stigma) yesaffron corolla inogadzirwa nekuora kwecarotene yakadai sezeaxanthin uye ine chimiro chakakosha. Iyo inonyanya kukosha safranal mu trimethylcyclethylene derivatives, inoverengera 50% yemafuta akazara anopisa. 72%, ndicho chigadzirwa chekudzikisira checrocin, uye zvakare imwe yemhando yekudzora zviratidzo zvechinyakare Chinese mushonga Zangsafflower. Dzimwe nyanzvi dzakaona makomisheni makumi mana nematanhatu kubva mumafuta esafuroni anopisa, anoverengera 46% yemafuta akazara. Pakati pavo, 90.99 ketone compounds inonzi 5%, 6.16 aldehyde compounds yakaverengerwa 5%, 2.39 alcohol compounds yakaverengerwa 6%, 4.98 acid compounds inonzi 6%, 19.77 olefin compounds inotora 8%, uye olefin yakasanganiswa oxides ye36.42 oxides. 2%, 5.74 alkane compounds akaverengera 8%, 12.5 ester compounds akaverengera 2%, uye 0.48 mamwe makomisheni akaverengera 4%. Pakati pezvakaonekwa zvinopisa zvemafuta zvikamu zvesafuroni, izvo zvine huwandu hwakanyanya zvakanyanya maolefin uye olefin oxides, ari terpenoid makomisheni. Mukuwedzera, izvo zvine huwandu hwehuwandu hwehuwandu huwandu hweasidhi.

2). Flavonoids Flavonoids inonyanya kugoverwa mu perianth yesafironi. Zvakajairika zvinosanganisira vetch glycoside, quercetin-3-p-coumaroylglucoside, kaempferol-3-glucose-6-acetylglucoside uye Kaempferol-3-glucose-glucoside, delphinidin, trimethyldelphinidin, nezvimwewo.

3). Volatile oiri precursors. Chikamu chemafuta anopisa anokonzeresa anogadzirwa nenzira dzakasiyana dzekushatisa panguva yekuomeswa uye kuchengetwa kwesaffron stigmas ndeye glycoside makomisheni e trimethylcyclohexene derivatives, kunyanya kusanganisira crocin uye zvichingodaro. Crocein ndiyo inonyanya kuvava chikamu musafuroni. Inogona kuchinjwa kuva safranal pasi pemamiriro ane acidic kana alkaline kana pasi pekuita kwema enzymes. Ichi ndichowo chikonzero nei zvinyorwa zvesafranal mumhando dzakasiyana zvakasiyana.

4). Conjugated polyenes uye glycosides yavo Conjugated polyenes uye glycosides avo ndiwo makuru ane mavara emukati mune yechinyakare Chinese mushonga safuroni. Inonyanya kusanganisira zvikamu zviviri zvinotevera: (1) Carotenoids uye glycosides Crocetin ndiyo chikamu chikuru che carotenoids uye glycosides yavo. Kusanganisira carotenoid crocetin uye glycosides ayo, akadai gentiobioside, glucoside, digentisic acid glycoside, gentioglucoside uye diglucoside; B-crocetin, C-crocetin, nezvimwewo (2) Carotenes inonyanya kusanganisira A uye B-carotene, yakadai se lycopene uye zeaxanthin.

5). Zvimwe zvinonyanya zvinosanganisira phenols, chitinase, triterpene saponins uye steroidal saponins.

4harmacological chiito

1). Mhedzisiro pachibereko cheSaffron inobvisa ine inonakidza mhedzisiro pane ese ari ega chibereko uye in vivo chibereko chembeva, guinea nguruve, tsuro, imbwa uye katsi. Chibereko chenhumbu chinowedzera kunzwa; kurongeka kwekusimba kwezvakasiyana-siyana zvesafranin zvinyorwa ndezvi: decoction> ethanol extract> volatile components> ether extract. Mhedzisiro yekunakidzwa kwechibereko inogona kuvharwa zvishoma ne ergotamine ethanesulfonate, iyo isinganzwisisike kune atropine. Nokudaro, zvinotendwa kuti chikamu chemugumisiro pachibereko chinokonzera zvakananga pane uterine myocytes, uye chikamu chine chokuita neadrenergic receptors.

2). Mhedzisiro painotenderera system Saffron inobvisa inogona kudzikisa BP yembwa nekatsi anesthetized kwenguva yakareba uye ine inonakidza mhedzisiro pakufema. Painoderedza BP, renal vhoriyamu inoderera, zvichiratidza renal vasoconstriction, uye anewo constrict mhedzisiro pamitsipa yeropa. Iyo ine yakakosha inhibitory mhedzisiro pamoyo wechuchi uri wega. Maererano nekuongorora kwemakemikari, zvikamu zvinodzivisa mwoyo zvine chokuita ne potassium munyu. Nokudaro, tsvakurudzo yezvemishonga yeramangwana pasafuroni inofanira kutanga yabvisa potassium munyu.

3). Anti-tumor effect Saffron gadziriro dzine pachena anti-bundu uye anti-cancer kugona, kunyanya safron inobvisa (dimethylcrocetin) pane leukemia, kenza ye ovarian, cancer cancer, rhabdomyosarcoma, colon cancer, papillosarcoma, uye flat cell bundu uye nyoro matishu sarcoma, nezvimwe. ose ane simba inhibitory effects. Iyo anti-cancer nzira inogona kunge iri yekuparadza iyo DNA synthase system, kureva, kuparadza iyo DNA-protein yekuonana nevamiriri senge topoisomerase II iyo yakakosha kune cellular DNA synthesis, nekudaro ichivharira synthesis yeDNA neRNA, nekudaro ichitadzisa kukura. ye tumor cell. effect. Mukuwedzera, macrocins anodzivisawo kushanda kwemasero eprotein kinases uye kutaura kweproto-oncogenes.

4). Mhedzisiro pachiropa uye gallbladder Saffron yakatorwa ine choleretic effect, uye yayo inoshanda zvinhu ndeye α-crocetin sodium munyu uye crocetin ester. α-Saffron acid inogona kuderedza cholesterol uye kuwedzera mafuta metabolism. Inogona kushandiswa nemishonga yechivanhu yechiChinese yakadai sehawthorn, cassia, uye Alisma kurapa chiropa chine mafuta.

5). Antioxidant effect Saffron inotorwa, kunyanya crocin, inogona kunyatso kuvharidzira kuita kweokisijeni isina radicals uye xanthine oxidase, ichiratidza antioxidant biological chiitiko.

6). Chengetedza itsvo. Nekudzidza rat C-BSA nephritis modhi, zvakaonekwa kuti proteinuria uye renal pathological kukuvara kwakaderedzwa mumakonzo muboka rekuyedza. Pakati pavo, safironi inonyanya kurambidza cyclooxygenase uye inoderedza kuumbwa kweprostaglandin, nekudaro kusunungura renal capillaries, kuwedzera kuyerera kweropa, uye kukurudzira kugadziriswa kwekukuvara kwekuzvimba. Zvinokurudzirwa kuti safironi inogona kukanganisa kuitika kwekuzvimba kwetsvo nekuvandudza kusunungurwa kweplatelet uye vamiririri vanopisa.

7). Kupindira mu arrhythmia Crocemic acid, iyo inoshandiswa mumucheka wesafuroni, ine simba rakanaka pane ventricular arrhythmia mienzaniso inokonzerwa neaconitine, ouabain uye calcium chloride, inopa miedzo yekushandiswa kwesafuroni mukurapa arrhythmia. Izvi zvinopa hwaro hwekuita kweimwe budiriro uye tsvakiridzo pasafuroni sechinyakare Chinese mushonga kugadzirira kurwisa arrhythmia uye myocardial ischemia, zvichiratidza kuti safironi inogona kunzi rudzi rutsva rwekudzivirira kwehutano-kutarisira echinyakare mushonga weChina wekudzivirira yemoyo uye cerebrovascular zvirwere.

8). Regulate immune function. Saffron inobvisa ine mhedzisiro yekusimudzira kutenderera kweropa uye kubvisa stasis yeropa, antibacterial uye anti-inflammatory, uyezve inosimudzira kutsungirira kwemuviri uye inowedzera zviri mukati memasero edziviriro, nekudaro inovandudza kusadzivirirwa kwemuviri, kudzora qi uye kufamba kweropa, uye kuenzanisa. muviri wemunhu. Basa reyin uye yang.

9). Kudzivirira uye kubata atherosclerosis. Saffron inobvisa ine simba rakanaka mukudzora lipids yeropa, kuderedza BP uye nokudaro kudzivirira nekurapa atherosclerosis.

10). Retinal protection: Tsuro chena dzekuNew Zealand dzakashandiswa kugadzira mhando yemhuka yehigh intraocular pressure. Imwe dhizimusi yesafuroni yakatorwa yakabayiwa kubva mutsinga yenzeve kamwe chete pazuva, uye boka rekudzora repamusoro rakamiswa. Zvigumisiro zvakaratidza kuti nhamba ye retinal ganglion masero muboka rekurapa yakanga yakakura kudarika iyo iri muboka repamusoro-soro (P <0.05), zvichiratidza kuti safroni yakatorwa yakavandudza retinal kutenderera kweropa uye yakavhara migumisiro yeischemia uye hypoxia pa retinal. ganglion masero ari pasi pechisingaperi chakakwira intraocular pressure mamiriro (RGC) kukuvadzwa uye kudzivirira RGC. Zvinokurudzirwa kuti safuroni inobviswa inogona kuchengetedza maRGCs nekudzikisa mahara radicals mu retina uye kuvhara mahara radical kukuvara kune membrane chimiro, subcellular organelles uye nuclei yeRGCs. 11. Mimwe migumisiro Saffron ethanol extract (CSE) inogona kudzivirira ethanol-induced inhibition yenguva refu potentiation (LPT) mu hippocampus. Mu serrated gyrus yemakonzo anesthetized, CSE (250 mg·kg-1) inogonawo kudzivirira zvinobudirira LPT inhibition inokonzerwa neacetaldehyde pasina kukanganisa basa rekudzidza remakonzo. Mvura yemvura yesafironi inogona kuvharidzira zvakanyanya kubereka huturu hunogadzirwa nemishonga inopesana nekenza yakadai se cisplatin, cyclophosphamide, mitomycin C uye urethan, nepo inhibiting Kukura kwechigumisiro kwakanga kusina kunyanya kuenderana nedosi. Izvi zvinonyanya kuitika nekuti safuroni yakatorwa inoderedza zvakanyanya mhedzisiro yekubereka chepfu pachiropa glutathione S-transferase (GST). Chimiro, kuravira uye kushanda zvakanaka: kutapira, kwazvakarerekera uye kusina chepfu. Inopinda mumoyo uye chiropa meridians. Inosimudzira kutenderera kweropa uye inobvisa stasis yeropa, inoparadzira kushushikana uye kuvhura mapfundo. Inogona kushandiswa kurapa kushushikana, chifuva uye diaphragm tightness, kurutsa ropa, typhoid fever, kutya uye kuona, amenorrhea muvakadzi, postpartum ropa stasis uye kurwadziwa mudumbu, uye kuzvimba uye kurwadziwa kubva pakudonha.

              

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